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8HQF

Crystal structure of SARS-Cov-2 main protease G15S mutant in complex with inhibitor YH-53

Summary for 8HQF
Entry DOI10.2210/pdb8hqf/pdb
DescriptorNon-structural protein 7, N-[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxidanylidene-3-[(3S)-2-oxidanylidenepyrrolidin-3-yl]propan-2-yl]amino]-4-methyl-1-oxidanylidene-pentan-2-yl]-4-methoxy-1H-indole-2-carboxamide (3 entities in total)
Functional Keywordsviral protein-inhibitor complex, viral protein/inhibitor
Biological sourceSevere acute respiratory syndrome coronavirus 2
Total number of polymer chains2
Total formula weight67509.07
Authors
Zeng, P.,Zhang, J.,Li, J. (deposition date: 2022-12-13, release date: 2024-01-31)
Primary citationZeng, P.,Zhang, J.,Li, J.
Crystal structure of SARS-Cov-2 main protease G15S mutant in complex with inhibitor YH-53
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.51 Å)
Structure validation

221051

數據於2024-06-12公開中

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