8CY2
CamA Adenine Methyltransferase Complexed to Cognate Substrate DNA and Inhibitor APNEA (Compound 9)
8CY2 の概要
エントリーDOI | 10.2210/pdb8cy2/pdb |
分子名称 | Site-specific DNA-methyltransferase (adenine-specific), DNA Strand 1, DNA Strand 2, ... (7 entities in total) |
機能のキーワード | dna adenine methylation, protein-dna complex, transferase, dna binding protein, dna binding protein-dna complex, dna binding protein/dna |
由来する生物種 | Clostridioides difficile 詳細 |
タンパク質・核酸の鎖数 | 9 |
化学式量合計 | 234266.82 |
構造登録者 | |
主引用文献 | Zhou, J.,Horton, J.R.,Menna, M.,Fiorentino, F.,Ren, R.,Yu, D.,Hajian, T.,Vedadi, M.,Mazzoccanti, G.,Ciogli, A.,Weinhold, E.,Huben, M.,Blumenthal, R.M.,Zhang, X.,Mai, A.,Rotili, D.,Cheng, X. Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile- Specific DNA Adenine Methyltransferase Required for Normal Sporulation and Persistence. J.Med.Chem., 66:934-950, 2023 Cited by PubMed: 36581322DOI: 10.1021/acs.jmedchem.2c01789 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.81 Å) |
構造検証レポート
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