8C8S
Crystal structure of human DNA cross-link repair 1A in complex with hydroxamic acid inhibitor (compound 21).
8C8S の概要
エントリーDOI | 10.2210/pdb8c8s/pdb |
分子名称 | DNA cross-link repair 1A protein, (2~{R})-3-[6-chloranyl-2-(prop-2-enylamino)quinazolin-4-yl]-2-methyl-~{N}-oxidanyl-propanamide, ZINC ION, ... (4 entities in total) |
機能のキーワード | exonuclease, snm1a, nuclease inhibition, hydrolase |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 39373.66 |
構造登録者 | Yosaatmadja, Y.,Newman, J.A.,Baddock, H.T.,Bielinski, M.,von Delft, F.,Bountra, C.,McHugh, P.J.,Schofield, C.J.,Gileadi, O. (登録日: 2023-01-20, 公開日: 2024-01-31) |
主引用文献 | Yosaatmadja, Y.,Newman, J.A.,Baddock, H.T.,Bielinski, M.,von Delft, F.,Bountra, C.,McHugh, P.J.,Schofield, C.J.,Gileadi, O. Crystal structure of human DNA cross-link repair 1A in complex with hydroxamic acid inhibitor (compound 21). To Be Published, |
実験手法 | X-RAY DIFFRACTION (1.8 Å) |
構造検証レポート
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