8C5Q

CK2 kinase bound to inhibitor AB668

Summary for 8C5Q

• Entry DOI: 10.2210/pdb8c5q/pdb
• Descriptor: Casein kinase II subunit alpha, SULFATE ION, 2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{H}-indole-2-carboxylate, ... (6 entities in total)
• Functional Keywords: kinase bivalent inhibitor, transferase
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 2
• Total formula weight: 88433.44

Authors

Krimm, I.,Guichou, J.F. (deposition date: 2023-01-10, release date: 2024-01-24)

• Primary citation: Krimm, I.,Guichou, J.F.; CK2 kinase bound to inhibitor AB668; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.5 Å)