8C11

BRD4 in complex with 2-(2-(4-(3,5-dimethylisoxazol-4-yl)-1H-pyrazol-1-yl)acetamido)-N-ethylpropanamide

Summary for 8C11

• Entry DOI: 10.2210/pdb8c11/pdb
• Descriptor: Bromodomain-containing protein 4, (2~{S})-2-[2-[4-(3,5-dimethyl-1,2-oxazol-4-yl)pyrazol-1-yl]ethanoylamino]-~{N}-ethyl-propanamide (3 entities in total)
• Functional Keywords: brd4, del, dels, inhibitor, dna encoded library, transcription
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 15679.03

Authors

Martin, M.P.,Noble, M.E.N. (deposition date: 2022-12-19, release date: 2023-12-27)

• Primary citation: Waring, M.J.; BRD4 complex with compound 22; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.8 Å)