8C11
BRD4 in complex with 2-(2-(4-(3,5-dimethylisoxazol-4-yl)-1H-pyrazol-1-yl)acetamido)-N-ethylpropanamide
Summary for 8C11
Entry DOI | 10.2210/pdb8c11/pdb |
Descriptor | Bromodomain-containing protein 4, (2~{S})-2-[2-[4-(3,5-dimethyl-1,2-oxazol-4-yl)pyrazol-1-yl]ethanoylamino]-~{N}-ethyl-propanamide (3 entities in total) |
Functional Keywords | brd4, del, dels, inhibitor, dna encoded library, transcription |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 15679.03 |
Authors | |
Primary citation | Waring, M.J. BRD4 complex with compound 22 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
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