7Z9V
Crystal structure of the C-terminal catalytic domain of Plasmodium falciparum CTP:phosphocholine cytidylyltransferase with 1,4-Anhydroerythritol
Summary for 7Z9V
Entry DOI | 10.2210/pdb7z9v/pdb |
Descriptor | Cholinephosphate cytidylyltransferase, Guanidinium, (3~{S},4~{R})-oxolane-3,4-diol, ... (4 entities in total) |
Functional Keywords | plasmodium falciparum cct inhibitors fragments, transferase |
Biological source | Plasmodium falciparum (malaria parasite P. falciparum) |
Total number of polymer chains | 1 |
Total formula weight | 21198.57 |
Authors | Duclovel, C.,Gelin, M.,Krimm, I.,Cerdan, R.,Guichou, J.-F. (deposition date: 2022-03-21, release date: 2023-03-29, Last modification date: 2024-02-07) |
Primary citation | Duclovel, C.,Gelin, M.,Wein, S.,Wengelnik, K.,Krimm, I.,Guichou, J.F.,Cerdan, R. Crystallographic screening using ultra-low-molecular-weight ligands to guide drug design of PfCCT inhibitors. To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
Download full validation report