7TTE
Tubulin-RB3_SLD in complex with compound 12j
7TTE の概要
エントリーDOI | 10.2210/pdb7tte/pdb |
分子名称 | Tubulin alpha-1B chain, Tubulin beta chain, Stathmin-4, ... (9 entities in total) |
機能のキーワード | microtubule inhibitor, colchicine, cell cycle, cancer, inhibitor complex, cell cycle-inhibitor complex, cell cycle/inhibitor |
由来する生物種 | Rattus norvegicus (Norway rat) 詳細 |
タンパク質・核酸の鎖数 | 5 |
化学式量合計 | 214832.77 |
構造登録者 | |
主引用文献 | Pochampally, S.,Hartman, K.L.,Wang, R.,Wang, J.,Yun, M.K.,Parmar, K.,Park, H.,Meibohm, B.,White, S.W.,Li, W.,Miller, D.D. Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo. Acs Pharmacol Transl Sci, 6:526-545, 2023 Cited by PubMed: 37082747DOI: 10.1021/acsptsci.2c00108 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.7 Å) |
構造検証レポート
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