7N03
Crystal structure of MTH1 in complex with compound 31
Summary for 7N03
Entry DOI | 10.2210/pdb7n03/pdb |
Descriptor | 7,8-dihydro-8-oxoguanine triphosphatase, 4-anilino-6-(hexylamino)-N-methylquinoline-3-carboxamide, SULFATE ION, ... (4 entities in total) |
Functional Keywords | inhibitor, hydrolase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 18684.21 |
Authors | Eron, S.J. (deposition date: 2021-05-24, release date: 2021-11-03, Last modification date: 2023-10-18) |
Primary citation | Veits, G.K.,Henderson, C.S.,Vogelaar, A.,Eron, S.J.,Lee, L.,Hart, A.,Deibler, R.W.,Baddour, J.,Elam, W.A.,Agafonov, R.V.,Freda, J.,Chaturvedi, P.,Ladd, B.,Carlson, M.W.,Vora, H.U.,Scott, T.G.,Tieu, T.,Jain, A.,Chen, C.L.,Kibbler, E.S.,Pop, M.S.,He, M.,Kern, G.,Maple, H.J.,Marsh, G.P.,Norley, M.C.,Oakes, C.S.,Henderson, J.A.,Sowa, M.E.,Phillips, A.J.,Proia, D.A.,Park, E.S.,Patel, J.S.,Fisher, S.L.,Nasveschuk, C.G.,Zeid, R. Development of an AchillesTAG degradation system and its application to control CAR-T activity Curr Res Chem Biol, 1:100010-, 2021 Cited by DOI: 10.1016/j.crchbi.2021.100010PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.13 Å) |
Structure validation
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