7F9R
Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in Complex with inhibitor L95, L-Proline and Febrifugine
Summary for 7F9R
Entry DOI | 10.2210/pdb7f9r/pdb |
Descriptor | Prolyl-tRNA synthetase (ProRS), ~{N}-[4-[(3~{S})-3-cyano-3-cyclopropyl-2-oxidanylidene-pyrrolidin-1-yl]-6-methyl-pyridin-2-yl]-2-phenyl-ethanamide, 3-{3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl}quinazolin-4(3H)-one, ... (7 entities in total) |
Functional Keywords | protein translation, inhibitor, prs, atp pocket, double drug, ligase, ligase-ligase inhibitor complex, ligase/ligase inhibitor |
Biological source | Toxoplasma gondii |
Total number of polymer chains | 1 |
Total formula weight | 59233.55 |
Authors | Manickam, Y.,Malhotra, N.,Sharma, A. (deposition date: 2021-07-04, release date: 2022-07-06, Last modification date: 2023-11-29) |
Primary citation | Malhotra, N.,Manickam, Y.,Sharma, A. TgPRS with double inhibitors To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.83 Å) |
Structure validation
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