7EHY

BRD4-BD1 in complex with LT-448-138

Summary for 7EHY

• Entry DOI: 10.2210/pdb7ehy/pdb
• Descriptor: Bromodomain-containing protein 4, 1-[2,4-dimethyl-5-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-pyrrol-3-yl]ethanone (3 entities in total)
• Functional Keywords: inhibitor, brd4, bd1, gene regulation
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15234.63

Authors

Zheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y. (deposition date: 2021-03-30, release date: 2022-03-30, Last modification date: 2023-11-29)

• Primary citation: Zheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y.; BRD4-BD1 in complex with LT-642-602; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.51 Å)