7DI7
Falcilysin in complex with chloroquine
Summary for 7DI7
Entry DOI | 10.2210/pdb7di7/pdb |
Descriptor | Falcilysin, ACETATE ION, N4-(7-CHLORO-QUINOLIN-4-YL)-N1,N1-DIETHYL-PENTANE-1,4-DIAMINE, ... (5 entities in total) |
Functional Keywords | protein binding-inhibitor complex, protein binding/inhibitor |
Biological source | Plasmodium falciparum 3D7 |
Total number of polymer chains | 1 |
Total formula weight | 135542.73 |
Authors | Lin, J.Q.,El Sahili, A.,Lescar, J. (deposition date: 2020-11-18, release date: 2021-12-01, Last modification date: 2024-05-29) |
Primary citation | Wirjanata, G.,Lin, J.,Dziekan, J.M.,El Sahili, A.,Chung, Z.,Tjia, S.,Binte Zulkifli, N.E.,Boentoro, J.,Tham, R.,Jia, L.S.,Go, K.D.,Yu, H.,Partridge, A.,Olsen, D.,Prabhu, N.,Sobota, R.M.,Nordlund, P.,Lescar, J.,Bozdech, Z. Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development. Cell Chem Biol, 31:743-759.e8, 2024 Cited by PubMed: 38593807DOI: 10.1016/j.chembiol.2024.03.002 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.82 Å) |
Structure validation
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