6Z5D
Crystal structure of haspin (GSG2) in complex with macrocycle ODS2004082
Summary for 6Z5D
Entry DOI | 10.2210/pdb6z5d/pdb |
Descriptor | Serine/threonine-protein kinase haspin, (4S)-2-METHYL-2,4-PENTANEDIOL, DIMETHYL SULFOXIDE, ... (7 entities in total) |
Functional Keywords | kinase, kinase inhibitor, haspin, gsg2 macrocycle, nanocyclic, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 41503.43 |
Authors | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-05-26, release date: 2020-06-03, Last modification date: 2024-01-24) |
Primary citation | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of haspin (GSG2) in complex with macrocycle ODS2004082 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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