6QXK
Human PIM1 bound to OX0999
Summary for 6QXK
Entry DOI | 10.2210/pdb6qxk/pdb |
Descriptor | Serine/threonine-protein kinase pim-1, Pimtide, 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one, ... (4 entities in total) |
Functional Keywords | kinase, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 37667.91 |
Authors | Alexander, L.T.,Elkins, J.M.,Russell, A.,Bountra, C.,Edwards, A.M.,Knapp, S. (deposition date: 2019-03-07, release date: 2019-04-24, Last modification date: 2024-01-24) |
Primary citation | Knapp, S.,Elkins, J.M.,Alexander, L.T.,Russell, A. PIM1 bound to OX0999 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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