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6QXK

Human PIM1 bound to OX0999

Summary for 6QXK
Entry DOI10.2210/pdb6qxk/pdb
DescriptorSerine/threonine-protein kinase pim-1, Pimtide, 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one, ... (4 entities in total)
Functional Keywordskinase, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight37667.91
Authors
Alexander, L.T.,Elkins, J.M.,Russell, A.,Bountra, C.,Edwards, A.M.,Knapp, S. (deposition date: 2019-03-07, release date: 2019-04-24, Last modification date: 2024-01-24)
Primary citationKnapp, S.,Elkins, J.M.,Alexander, L.T.,Russell, A.
PIM1 bound to OX0999
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

218853

数据于2024-04-24公开中

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