6KYA
Crystal structure of human TLR8 in complex TH1027
6KYA の概要
エントリーDOI | 10.2210/pdb6kya/pdb |
分子名称 | Toll-like receptor 8, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total) |
機能のキーワード | immune system |
由来する生物種 | Homo sapiens (Human) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 192191.03 |
構造登録者 | |
主引用文献 | Jiang, S.,Tanji, H.,Yin, K.,Zhang, S.,Sakaniwa, K.,Huang, J.,Yang, Y.,Li, J.,Ohto, U.,Shimizu, T.,Yin, H. Rationally Designed Small-Molecule Inhibitors Targeting an Unconventional Pocket on the TLR8 Protein-Protein Interface. J.Med.Chem., 63:4117-4132, 2020 Cited by PubMed: 32233366DOI: 10.1021/acs.jmedchem.9b02128 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.89 Å) |
構造検証レポート
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