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6KE0

Crystal structure of PDE10A in complex with a triazolopyrimidine inhibitor

Summary for 6KE0
Entry DOI10.2210/pdb6ke0/pdb
Related6KDX 6KDZ
DescriptorcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A, ZINC ION, MAGNESIUM ION, ... (4 entities in total)
Functional Keywordsinhibitor, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight79753.69
Authors
Amano, Y.,Honbou, K. (deposition date: 2019-07-03, release date: 2019-08-14, Last modification date: 2023-11-22)
Primary citationChino, A.,Honda, S.,Morita, M.,Yonezawa, K.,Hamaguchi, W.,Amano, Y.,Moriguchi, H.,Yamazaki, M.,Aota, M.,Tomishima, M.,Masuda, N.
Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors.
Bioorg.Med.Chem., 27:3692-3706, 2019
Cited by
PubMed: 31301949
DOI: 10.1016/j.bmc.2019.07.010
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.95 Å)
Structure validation

217705

数据于2024-03-27公开中

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