6K1Q
Human endothelin receptor type-B in complex with inverse agonist IRL2500
Summary for 6K1Q
Entry DOI | 10.2210/pdb6k1q/pdb |
Descriptor | Endothelin B receptor,Endolysin,Endothelin B receptor, (2~{S})-2-[[(2~{R})-2-[(3,5-dimethylphenyl)carbonyl-methyl-amino]-3-(4-phenylphenyl)propanoyl]amino]-3-(1~{H}-indol-3-yl)propanoic acid, PHOSPHATE ION, ... (5 entities in total) |
Functional Keywords | alpha helical, signaling protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 1 |
Total formula weight | 55933.97 |
Authors | |
Primary citation | Nagiri, C.,Shihoya, W.,Inoue, A.,Kadji, F.M.N.,Aoki, J.,Nureki, O. Crystal structure of human endothelin ETBreceptor in complex with peptide inverse agonist IRL2500. Commun Biol, 2:236-236, 2019 Cited by PubMed: 31263780DOI: 10.1038/s42003-019-0482-7 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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