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6JJ6

BRD4 in complex with 500

Summary for 6JJ6
Entry DOI10.2210/pdb6jj6/pdb
DescriptorBromodomain-containing protein 4, 1-methyl-6-(3-(4-methylpiperazine-1-carbonyl)benzyl)-1,2a1,5a,6-tetrahydro-2H-pyrido[3',2':6,7]azepino[4,3,2-cd]isoindol-2-one (3 entities in total)
Functional Keywordsbrd4, inhibitor, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15348.73
Authors
Xu, J.,Chen, Y.,Jiang, F.,Zhu, J. (deposition date: 2019-02-25, release date: 2020-02-26, Last modification date: 2024-03-27)
Primary citationXu, J.,Zhu, J.,Chen, Y.,Jiang, F.
BRD4 in complex with ZZM1
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.4 Å)
Structure validation

218500

건을2024-04-17부터공개중

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