6HRO
Crystal structure of Ebolavirus glycoprotein in complex with inhibitor 118a
6HRO の概要
エントリーDOI | 10.2210/pdb6hro/pdb |
分子名称 | Envelope glycoprotein,Envelope glycoprotein,Envelope glycoprotein, Envelope glycoprotein, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (8 entities in total) |
機能のキーワード | ebola glycoprotein, structure-based in silico screening, 118a, natural compound, viral protein |
由来する生物種 | Zaire ebolavirus (strain Mayinga-76) (ZEBOV) 詳細 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 58685.43 |
構造登録者 | |
主引用文献 | Shaikh, F.,Zhao, Y.,Alvarez, L.,Iliopoulou, M.,Lohans, C.,Schofield, C.J.,Padilla-Parra, S.,Siu, S.W.I.,Fry, E.E.,Ren, J.,Stuart, D.I. Structure-Based in Silico Screening Identifies a Potent Ebolavirus Inhibitor from a Traditional Chinese Medicine Library. J.Med.Chem., 62:2928-2937, 2019 Cited by PubMed: 30785281DOI: 10.1021/acs.jmedchem.8b01328 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.3 Å) |
構造検証レポート
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