6F5U
CRYSTAL STRUCTURE OF EBOLAVIRUS GLYCOPROTEIN IN COMPLEX WITH BEPRIDIL
6F5U の概要
エントリーDOI | 10.2210/pdb6f5u/pdb |
分子名称 | Envelope glycoprotein,Envelope glycoprotein,GP1, Envelope glycoprotein, alpha-D-mannopyranose-(1-6)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (8 entities in total) |
機能のキーワード | ebola virus, filoviridae, envelope glycoprotein, protein inhibitor complex, ibuprofen, benztropine, bepridil, paroxetine and sertraline, toremifene, viral protein |
由来する生物種 | Zaire ebolavirus (strain Mayinga-76) (ZEBOV) 詳細 |
細胞内の位置 | GP2: Virion membrane ; Single-pass type I membrane protein . GP1: Virion membrane ; Peripheral membrane protein. GP2-delta: Secreted : Q05320 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 57245.68 |
構造登録者 | |
主引用文献 | Ren, J.,Zhao, Y.,Fry, E.E.,Stuart, D.I. Target Identification and Mode of Action of Four Chemically Divergent Drugs against Ebolavirus Infection. J. Med. Chem., 61:724-733, 2018 Cited by PubMed: 29272110DOI: 10.1021/acs.jmedchem.7b01249 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.07 Å) |
構造検証レポート
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