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6EAS

Co-crystal of pseudokinase DRIK1 (drought responsive inactive kinase 1) bound to ENMD-2076

Summary for 6EAS
Entry DOI10.2210/pdb6eas/pdb
Descriptordrought responsive inactive kinase 1, 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine, GLYCEROL, ... (4 entities in total)
Functional Keywordsreceptor-like kinase, pseudokinase, maize, enmd-2076, structural genomics consortium, transferase-transferase inhibitor complex, sgc, transferase/transferase inhibitor
Biological sourceZea mays (Maize)
Total number of polymer chains1
Total formula weight35253.17
Authors
Aquino, B.,Counago, R.M.,Fala, A.M.,Massirer, K.B.,Elkins, J.M.,Arruda, P.,Structural Genomics Consortium (SGC) (deposition date: 2018-08-03, release date: 2018-08-22, Last modification date: 2023-10-11)
Primary citationAquino, B.,Counago, R.M.,Fala, A.M.,Massirer, K.B.,Elkins, J.M.,Arruda, P.
Co-crystal of pseudokinase DRIK1 with ENMD-2076
To be Published,
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

220472

数据于2024-05-29公开中

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