5Z90
BRD4 Bromodomain 1 with an inhibitor
Summary for 5Z90
| Entry DOI | 10.2210/pdb5z90/pdb |
| Descriptor | Bromodomain-containing protein 4, 1-ethyl-6-pyrrolidin-1-ylsulfonyl-benzo[cd]indol-2-one (3 entities in total) |
| Functional Keywords | brd4 bromodomain 1, inhibitor, complex, transcription-inhibitor complex, transcription/inhibitor |
| Biological source | Homo sapiens (Human) |
| Total number of polymer chains | 1 |
| Total formula weight | 15429.78 |
| Authors | |
| Primary citation | Xiao, S.,Chen, S.,Chen, H. BRD4 Bromodomain 1 with an inhibitor To Be Published, |
| Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
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