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5XXG

Crystal structure of SmyD3 in complex with covalent inhibitor 2

Summary for 5XXG
Entry DOI10.2210/pdb5xxg/pdb
DescriptorSMYD3, propyl 4-(4-chloranyl-2-phenyl-quinolin-7-yl)carbonylpiperazine-1-carboxylate, S-ADENOSYLMETHIONINE, ... (5 entities in total)
Functional Keywordsmethyltransferase, covalent inhibitor, smyd3, transferase, transferase-inhibitor complex, transferase/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight49635.04
Authors
Baburajendran, N.,Jansson, E.A. (deposition date: 2017-07-03, release date: 2018-08-08)
Primary citationBaburajendran, N.,Jansson, E.A.
Crystal structure of SmyD3 in complex with covalent inhibitor 2
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.14 Å)
Structure validation

221051

数据于2024-06-12公开中

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