5XHY
BRD4 bound with compound Bdi1
Summary for 5XHY
Entry DOI | 10.2210/pdb5xhy/pdb |
Descriptor | Bromodomain-containing protein 4, ~{N}-(4-cyclopropyl-1,3,3-trimethyl-2-oxidanylidene-quinoxalin-6-yl)-4-methyl-benzenesulfonamide (3 entities in total) |
Functional Keywords | chromatin regulator, transcription-inhibitor complex, transcription/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: O60885 |
Total number of polymer chains | 1 |
Total formula weight | 15153.58 |
Authors | |
Primary citation | Bing, X. BRD4 bound with compound Bdi1 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.976 Å) |
Structure validation
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