5WII
TraE protein in complex with 2-Chloroisonicotinic Acid
Summary for 5WII
Entry DOI | 10.2210/pdb5wii/pdb |
Descriptor | Conjugal transfer protein, 2-chloropyridine-4-carboxylic acid (3 entities in total) |
Functional Keywords | type iv secretion system, fragment-based drug design, complex, inhibitor, antimicrobial resistance, bacterial secretion, virb, protein transport |
Biological source | Escherichia coli |
Total number of polymer chains | 4 |
Total formula weight | 75429.97 |
Authors | Casu, B.,Arya, T.,Bessette, B.,Baron, C. (deposition date: 2017-07-19, release date: 2017-11-15, Last modification date: 2023-10-04) |
Primary citation | Casu, B.,Arya, T.,Bessette, B.,Baron, C. Fragment-based screening identifies novel targets for inhibitors of conjugative transfer of antimicrobial resistance by plasmid pKM101. Sci Rep, 7:14907-14907, 2017 Cited by PubMed: 29097752DOI: 10.1038/s41598-017-14953-1 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.79 Å) |
Structure validation
Download full validation report