5U44
Human PPARdelta ligand-binding domain in complexed with specific agonist 13
Summary for 5U44
Entry DOI | 10.2210/pdb5u44/pdb |
Related | 5U3Q 5U3R 5U3S 5U3T 5U3U 5U3V 5U3W 5U3X 5U3Y 5U3Z 5U40 5U41 5U42 5U43 5U45 5U46 |
Descriptor | Peroxisome proliferator-activated receptor delta, heptyl beta-D-glucopyranoside, S-1,2-PROPANEDIOL, ... (5 entities in total) |
Functional Keywords | ppardelta, ligand-binding domain, agonist, protein binding-activator complex, protein binding/activator |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 63964.42 |
Authors | Wu, C.-C.,Baiga, T.J.,Downes, M.,La Clair, J.J.,Atkins, A.R.,Richard, S.B.,Stockley-Noel, T.A.,Bowman, M.E.,Evans, R.M.,Noel, J.P. (deposition date: 2016-12-03, release date: 2017-03-22, Last modification date: 2023-10-04) |
Primary citation | Wu, C.C.,Baiga, T.J.,Downes, M.,La Clair, J.J.,Atkins, A.R.,Richard, S.B.,Fan, W.,Stockley-Noel, T.A.,Bowman, M.E.,Noel, J.P.,Evans, R.M. Structural basis for specific ligation of the peroxisome proliferator-activated receptor delta. Proc. Natl. Acad. Sci. U.S.A., 114:E2563-E2570, 2017 Cited by PubMed: 28320959DOI: 10.1073/pnas.1621513114 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.15 Å) |
Structure validation
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