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5R4X

XChem fragment screen -- CRYSTAL STRUCTURE OF THE BROMODOMAIN OF THE HUMAN ATAD2 in complex with N13413a

5R4X の概要
エントリーDOI10.2210/pdb5r4x/pdb
Group depositionXChem fragment screen (G_1002130)
分子名称ATPase family AAA domain-containing protein 2, 4-acetyl-N-ethylpiperazine-1-carboxamide, SULFATE ION, ... (5 entities in total)
機能のキーワードpandda, sgc - diamond i04-1 fragment screening, xchemexplorer, atpase family, aaa domain containing 2, ancca, aaa+ nuclear coregulator cancer-associated pro2000 protein, two aaa domain containing protein, sgc, structural genomics consortium, atp-binding, bromodomain, nucleotide-binding, phosphoprotein, signaling protein, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
由来する生物種Homo sapiens (Human)
タンパク質・核酸の鎖数1
化学式量合計16152.21
構造登録者
主引用文献Talon, R.,Krojer, T.,Fairhead, M.,Sethi, R.,Bradley, A.R.,Aimon, A.,Collins, P.,Brandao-Neto, J.,Douangamath, A.,Wright, N.,MacLean, E.,Zhang, R.,Dias, A.,Brennan, P.E.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.,von Delft, F.
XChem fragment screen
To Be Published,
実験手法
X-RAY DIFFRACTION (1.4 Å)
構造検証レポート
Validation report summary of 5r4x
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-07-17に公開中

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