5QR2
PanDDA analysis group deposition -- Crystal Structure of human ALAS2A in complex with Z1348371854
Summary for 5QR2
Entry DOI | 10.2210/pdb5qr2/pdb |
Group deposition | PanDDA analysis group deposition (G_1002078) |
Descriptor | 5-aminolevulinate synthase, erythroid-specific, mitochondrial, PYRIDOXAL-5'-PHOSPHATE, 5-(1,4-oxazepan-4-yl)pyridine-2-carbonitrile, ... (4 entities in total) |
Functional Keywords | sgc - diamond i04-1 fragment screening, pandda, xchemexplorer, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 105198.63 |
Authors | Bezerra, G.A.,Foster, W.,Bailey, H.,Shrestha, L.,Krojer, T.,Talon, R.,Brandao-Neto, J.,Douangamath, A.,Nicola, B.B.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.,Bountra, C.,Brennan, P.E.,Yue, W.W. (deposition date: 2019-05-22, release date: 2019-08-07, Last modification date: 2024-03-06) |
Primary citation | Bezerra, G.A.,Foster, W.,Bailey, H.,Shrestha, L.,Krojer, T.,Talon, R.,Brandao-Neto, J.,Douangamath, A.,Nicola, B.B.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.,Bountra, C.,Brennan, P.E.,Yue, W.W. PanDDA analysis group deposition To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.66 Å) |
Structure validation
Download full validation report