4YCM
Crystal structure of the calcium pump with bound marine macrolide BLS
Summary for 4YCM
Entry DOI | 10.2210/pdb4ycm/pdb |
Related | 4YCN |
Descriptor | Sarcoplasmic/endoplasmic reticulum calcium ATPase 1, SODIUM ION, SULFATE ION, ... (5 entities in total) |
Functional Keywords | membrane protein, p-type atpase, had fold, ca2+, ion pump, hydrolase |
Biological source | Oryctolagus cuniculus (Rabbit) |
Total number of polymer chains | 1 |
Total formula weight | 111932.58 |
Authors | Morita, M.,Ogawa, H.,Ohno, O.,Yamori, T.,Suenaga, K.,Toyoshima, C. (deposition date: 2015-02-20, release date: 2016-01-13, Last modification date: 2020-02-05) |
Primary citation | Morita, M.,Ogawa, H.,Ohno, O.,Yamori, T.,Suenaga, K.,Toyoshima, C. Biselyngbyasides, cytotoxic marine macrolides, are novel and potent inhibitors of the Ca(2+) pumps with a unique mode of binding Febs Lett., 589:1406-1411, 2015 Cited by PubMed: 25957767DOI: 10.1016/j.febslet.2015.04.056 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.2 Å) |
Structure validation
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