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4W4V

JNK2/3 in complex with 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(2-methylpyridin-4-yl)benzamide

Summary for 4W4V
Entry DOI10.2210/pdb4w4v/pdb
Related4W4W 4W4X 4W4Y
Descriptorc-Jun N-terminal kinase 3, 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(2-methylpyridin-4-yl)benzamide (3 entities in total)
Functional Keywordsjnk, map kinase, isoform selective, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight42708.83
Authors
Park, H.,Iqbal, S.,Hernandez, P.,Mora, R.,Zheng, K.,Feng, Y.,LoGrasso, P. (deposition date: 2014-08-15, release date: 2015-02-11, Last modification date: 2023-12-27)
Primary citationPark, H.,Iqbal, S.,Hernandez, P.,Mora, R.,Zheng, K.,Feng, Y.,LoGrasso, P.
Structural Basis and Biological Consequences for JNK2/3 Isoform Selective Aminopyrazoles.
Sci Rep, 5:8047-8047, 2015
Cited by
PubMed: 25623238
DOI: 10.1038/srep08047
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.01 Å)
Structure validation

217705

数据于2024-03-27公开中

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