4QIB
Oxidation-Mediated Inhibition of the Peptidyl-Prolyl Isomerase Pin1
Summary for 4QIB
Entry DOI | 10.2210/pdb4qib/pdb |
Descriptor | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, SULFATE ION, ... (4 entities in total) |
Functional Keywords | cis-trans isomerization, oxidation of active site cysteine, cysteine sulfenic-sulfinic acid redox regulation, parvulin, isomerase |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: Q13526 |
Total number of polymer chains | 1 |
Total formula weight | 18379.24 |
Authors | Innes, B.T.,Sowole, M.A.,Konermann, L.,Litchfield, D.W.,Brandl, C.J.,Shilton, B.H. (deposition date: 2014-05-30, release date: 2015-02-04, Last modification date: 2015-03-04) |
Primary citation | Innes, B.T.,Sowole, M.A.,Gyenis, L.,Dubinsky, M.,Konermann, L.,Litchfield, D.W.,Brandl, C.J.,Shilton, B.H. Peroxide-mediated oxidation and inhibition of the peptidyl-prolyl isomerase Pin1. Biochim.Biophys.Acta, 1852:905-912, 2015 Cited by PubMed: 25595659DOI: 10.1016/j.bbadis.2014.12.025 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.865 Å) |
Structure validation
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