4FIV
FIV PROTEASE COMPLEXED WITH AN INHIBITOR LP-130
4FIV の概要
エントリーDOI | 10.2210/pdb4fiv/pdb |
分子名称 | FELINE IMMUNODEFICIENCY VIRUS PROTEASE, 4-[2-(2-ACETYLAMINO-3-NAPHTALEN-1-YL-PROPIONYLAMINO)-4-METHYL-PENTANOYLAMINO]-3-HYDROXY-6-METHYL-HEPTANOIC ACID [1-(1-CARBAMOYL-2-NAPHTHALEN-1-YL-ETHYLCARBAMOYL)-PROPYL]-AMIDE (3 entities in total) |
機能のキーワード | aspartic protease, fiv, retropepsin, retrovirus, cat |
由来する生物種 | Feline immunodeficiency virus |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 13637.80 |
構造登録者 | Kervinen, J.,Lubkowski, J.,Zdanov, A.,Wlodawer, A.,Gustchina, A. (登録日: 1998-07-15, 公開日: 1999-01-13, 最終更新日: 2023-08-09) |
主引用文献 | Kervinen, J.,Lubkowski, J.,Zdanov, A.,Bhatt, D.,Dunn, B.M.,Hui, K.Y.,Powell, D.J.,Kay, J.,Wlodawer, A.,Gustchina, A. Toward a universal inhibitor of retroviral proteases: comparative analysis of the interactions of LP-130 complexed with proteases from HIV-1, FIV, and EIAV. Protein Sci., 7:2314-2323, 1998 Cited by PubMed: 9827997主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.8 Å) |
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