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3VFH

BlaC E166A CDC-1 Acyl-Intermediate

Summary for 3VFH
Entry DOI10.2210/pdb3vfh/pdb
Related3VFF 4EBI 4EBL 4EBM 4EBN 4EBO 4EBP
DescriptorBeta-lactamase, PHOSPHATE ION, (2R)-5-methylidene-2-{(1R)-2-oxo-1-[(phenylacetyl)amino]ethyl}-5,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, ... (4 entities in total)
Functional Keywordsbeta-lactamase, serine hydrolase, serine esterase, acyl-intermediate, hydrolase-hydrolase inhibitor complex, structural genomics, tb structural genomics consortium, tbsgc, hydrolase/hydrolase inhibitor
Biological sourceMycobacterium tuberculosis
Cellular locationCell membrane; Lipid-anchor (Potential): P0C5C1
Total number of polymer chains4
Total formula weight123285.84
Authors
Mire, J.A.,Sacchettini, J.C.,TB Structural Genomics Consortium (TBSGC) (deposition date: 2012-01-09, release date: 2012-09-19, Last modification date: 2023-09-13)
Primary citationXie, H.,Mire, J.A.,Kong, Y.,Chang, M.,Sacchettini, J.C.,Cirillo, J.D.,Rao, J.
BlaC-Specific Fluorogenic Probes for Rapid Tuberculosis Detection
To be Published,
Experimental method
X-RAY DIFFRACTION (2.57 Å)
Structure validation

217705

数据于2024-03-27公开中

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