3MA6
Crystal structure of kinase domain of TgCDPK1 in presence of 3BrB-PP1
3MA6 の概要
エントリーDOI | 10.2210/pdb3ma6/pdb |
分子名称 | Calmodulin-domain protein kinase 1, 3-(3-bromobenzyl)-1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine (3 entities in total) |
機能のキーワード | cdpk, parasitology, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, structural genomics, structural genomics consortium, sgc |
由来する生物種 | Toxoplasma gondii |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 69870.18 |
構造登録者 | Wernimont, A.K.,Qiu, W.,Amani, M.,Artz, J.D.,Hassani, A.A.,Senisterra, G.,Vedadi, M.,Sibley, L.D.,Lourido, S.,Shokat, K.,Zhang, C.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Weigelt, J.,Bochkarev, A.,Hui, R.,Lin, Y.H.,Structural Genomics Consortium (SGC) (登録日: 2010-03-23, 公開日: 2010-07-21, 最終更新日: 2017-11-08) |
主引用文献 | Wernimont, A.K.,Qiu, W.,Amani, M.,Artz, J.D.,Hassani, A.A.,Senisterra, G.,Vedadi, M.,Sibley, L.D.,Lourido, S.,Shokat, K.,Zhang, C.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Weigelt, J.,Bochkarev, A.,Hui, R.,Lin, Y.H. Crystal structure of kinase domain of TgCDPK1 in presence of 3BrB-PP1 To be Published, |
実験手法 | X-RAY DIFFRACTION (2.5 Å) |
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