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3MA6

Crystal structure of kinase domain of TgCDPK1 in presence of 3BrB-PP1

3MA6 の概要
エントリーDOI10.2210/pdb3ma6/pdb
分子名称Calmodulin-domain protein kinase 1, 3-(3-bromobenzyl)-1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine (3 entities in total)
機能のキーワードcdpk, parasitology, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, structural genomics, structural genomics consortium, sgc
由来する生物種Toxoplasma gondii
タンパク質・核酸の鎖数2
化学式量合計69870.18
構造登録者
主引用文献Wernimont, A.K.,Qiu, W.,Amani, M.,Artz, J.D.,Hassani, A.A.,Senisterra, G.,Vedadi, M.,Sibley, L.D.,Lourido, S.,Shokat, K.,Zhang, C.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Weigelt, J.,Bochkarev, A.,Hui, R.,Lin, Y.H.
Crystal structure of kinase domain of TgCDPK1 in presence of 3BrB-PP1
To be Published,
実験手法
X-RAY DIFFRACTION (2.5 Å)
構造検証レポート
Validation report summary of 3ma6
検証レポート(詳細版)ダウンロードをダウンロード

246905

件を2025-12-31に公開中

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