3IQ7
Crystal Structure of human Haspin in complex with 5-Iodotubercidin
3IQ7 の概要
エントリーDOI | 10.2210/pdb3iq7/pdb |
分子名称 | Serine/threonine-protein kinase haspin, PHOSPHATE ION, (2R,3R,4S,5R)-2-(4-AMINO-5-IODO-7H-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-(HYDROXYMETHYL)TETRAHYDROFURAN-3,4-DIOL, ... (6 entities in total) |
機能のキーワード | haspin, germ cell associated 2, haploid germ cell specific nuclear protein kinase, sgc, structural genomics consortium, atp-binding, cell cycle, chromatin regulator, kinase, magnesium, nucleotide-binding, nucleus, phosphoprotein, serine/threonine-protein kinase, transferase |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Nucleus: Q8TF76 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 41449.64 |
構造登録者 | Filippakopoulos, P.,Eswaran, J.,Keates, T.,Burgess-Brown, N.,Fedorov, O.,Pike, A.C.W.,Von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2009-08-19, 公開日: 2009-09-08, 最終更新日: 2023-11-01) |
主引用文献 | Eswaran, J.,Patnaik, D.,Filippakopoulos, P.,Wang, F.,Stein, R.L.,Murray, J.W.,Higgins, J.M.,Knapp, S. Structure and functional characterization of the atypical human kinase haspin. Proc.Natl.Acad.Sci.USA, 106:20198-20203, 2009 Cited by PubMed: 19918057DOI: 10.1073/pnas.0901989106 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2 Å) |
構造検証レポート
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