3AW1
Structure of SARS 3CL protease auto-proteolysis resistant mutant in the absent of inhibitor
3AW1 の概要
エントリーDOI | 10.2210/pdb3aw1/pdb |
関連するPDBエントリー | 3AVZ 3AW0 |
分子名称 | 3C-Like Proteinase (2 entities in total) |
機能のキーワード | hydrolase proteinase converting, hydrolase |
由来する生物種 | SARS coronavirus (SARS-CoV) |
細胞内の位置 | Non-structural protein 3: Host membrane; Multi-pass membrane protein (Potential). Non-structural protein 4: Host membrane; Multi-pass membrane protein (Potential). Non-structural protein 6: Host membrane; Multi-pass membrane protein (Potential). Non-structural protein 7: Host cytoplasm, host perinuclear region (By similarity). Non-structural protein 8: Host cytoplasm, host perinuclear region (By similarity). Non-structural protein 9: Host cytoplasm, host perinuclear region (By similarity). Non-structural protein 10: Host cytoplasm, host perinuclear region (By similarity): P0C6U8 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 67665.20 |
構造登録者 | Akaji, K.,Konno, H.,Mitsui, H.,Teruya, K.,Hattori, Y.,Ozaki, T.,Kusunoki, M.,Sanjho, A. (登録日: 2011-03-09, 公開日: 2011-12-14, 最終更新日: 2023-11-01) |
主引用文献 | Akaji, K.,Konno, H.,Mitsui, H.,Teruya, K.,Shimamoto, Y.,Hattori, Y.,Ozaki, T.,Kusunoki, M.,Sanjoh, A. Structure-Based Design, Synthesis, and Evaluation of Peptide-Mimetic SARS 3CL Protease Inhibitors. J.Med.Chem., 54:7962-7973, 2011 Cited by PubMed: 22014094DOI: 10.1021/jm200870n 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード