3AMV
ALLOSTERIC INHIBITION OF GLYCOGEN PHOSPHORYLASE A BY A POTENTIAL ANTIDIABETIC DRUG
3AMV の概要
エントリーDOI | 10.2210/pdb3amv/pdb |
分子名称 | PROTEIN (GLYCOGEN PHOSPHORYLASE), alpha-D-glucopyranose, PYRIDOXAL-5'-PHOSPHATE, ... (6 entities in total) |
機能のキーワード | diabetes, glycogen metabolism, phosphorylase a, inhibition, allosteric site, transferase |
由来する生物種 | Oryctolagus cuniculus (rabbit) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 98297.41 |
構造登録者 | Oikonomakos, N.G.,Tsitsanou, K.E.,Zographos, S.E.,Skamnaki, V.T. (登録日: 1999-02-18, 公開日: 1999-02-26, 最終更新日: 2023-12-27) |
主引用文献 | Oikonomakos, N.G.,Tsitsanou, K.E.,Zographos, S.E.,Skamnaki, V.T.,Goldmann, S.,Bischoff, H. Allosteric inhibition of glycogen phosphorylase a by the potential antidiabetic drug 3-isopropyl 4-(2-chlorophenyl)-1,4-dihydro-1-ethyl-2-methyl-pyridine-3,5,6-tricarbo xylate. Protein Sci., 8:1930-1945, 1999 Cited by PubMed: 10548038主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.1 Å) |
構造検証レポート
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