3A7E
Crystal structure of human COMT complexed with SAM and 3,5-dinitrocatechol
3A7E の概要
エントリーDOI | 10.2210/pdb3a7e/pdb |
関連するPDBエントリー | 1VID 3A7D 3BWM 3BWY |
分子名称 | Catechol O-methyltransferase, MAGNESIUM ION, S-ADENOSYLMETHIONINE, ... (5 entities in total) |
機能のキーワード | comt, alternative initiation, catecholamine metabolism, magnesium, methyltransferase, neurotransmitter degradation, s-adenosyl-l-methionine, transferase, cell membrane, membrane, metal-binding, phosphoprotein, signal-anchor, transmembrane |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Isoform Soluble: Cytoplasm. Isoform Membrane-bound: Cell membrane; Single-pass type II membrane protein; Extracellular side : P21964 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 24649.45 |
構造登録者 | |
主引用文献 | Nonaka, Y.,Momose, T.,Ozawa, T.,Ozawa, M.,Nakatsu, M.,Tsuji, E.,Okazaki, K.,Takase, Y.,Kiyotani, T. Hit to Lead: Comprehensive Strategy of de novo Scaffold Generation by FBDD. Part 1: In silico Fragments Linking and Verification of Spatial Proximity using Inter Ligand NOE Approachs To be Published, |
実験手法 | X-RAY DIFFRACTION (2.8 Å) |
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