2W4O
Crystal structure of Human CAMK4 in complex with 4-Amino(sulfamoyl- phenylamino)-triazole-carbothioic acid (2,6-difluoro-phenyl)-amide)
2W4O の概要
エントリーDOI | 10.2210/pdb2w4o/pdb |
分子名称 | CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE IV, 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE (3 entities in total) |
機能のキーワード | calmodulin-binding, nucleotide-binding, serine/threonine-protein kinase, atp-binding, phosphoprotein, kinase, nucleus, transferase |
由来する生物種 | HOMO SAPIENS (HUMAN) |
細胞内の位置 | Cytoplasm: Q16566 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 39751.72 |
構造登録者 | Muniz, J.R.C.,Rellos, P.,Gileadi, O.,Fedorov, O.,Filippakopoulos, P.,Salah, E.,Pike, A.,Phillips, C.,Niesen, F.,Shrestha, L.,Burgess-Brown, N.,Bullock, A.,Berridge, G.,von Delft, F.,Edwards, A.M.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Knapp, S. (登録日: 2008-11-28, 公開日: 2009-01-20, 最終更新日: 2024-02-07) |
主引用文献 | Muniz, J.R.C.,Rellos, P.,Gileadi, O.,Fedorov, O.,Filippakopoulos, P.,Salah, E.,Pike, A.,Phillips, C.,Niesen, F.,Shrestha, L.,Burgess-Brown, N.,Bullock, A.,Berridge, G.,von Delft, F.,Edwards, A.M.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Knapp, S. Crystal Structure of Human Camk4 in Complex with 4-Amino(Sulfamoyl-Phenylamino)-Triazole- Carbothioic Acid (2,6-Difluoro-Phenyl)-Amide) To be Published, |
実験手法 | X-RAY DIFFRACTION (2.17 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード