2W0V
Crystal structure of Glmu from Haemophilus influenzae in complex with quinazoline inhibitor 1
2W0V の概要
エントリーDOI | 10.2210/pdb2w0v/pdb |
関連するPDBエントリー | 2V0H 2V0I 2V0J 2V0K 2V0L 2VD4 2W0W |
分子名称 | GLUCOSAMINE-1-PHOSPHATE N-ACETYLTRANSFERASE, 6-(CYCLOPROP-2-EN-1-YLMETHOXY)-2-[6-(CYCLOPROPYLMETHYL)-5-OXO-3,4,5,6-TETRAHYDRO-2,6-NAPHTHYRIDIN-2(1H)-YL]-7-METHOXYQUINAZOLIN-4(3H)-ONE, TETRAETHYLENE GLYCOL, ... (6 entities in total) |
機能のキーワード | peptidoglycan synthesis, glmu, bacterial, inhibitor, magnesium, cell shape, transferase, active site, metal-binding, cell wall biogenesis/degradation, multifunctional enzyme, nucleotidyltransferase, acyltransferase, uridyltransferase |
由来する生物種 | HAEMOPHILUS INFLUENZAE |
細胞内の位置 | Cytoplasm (By similarity): P43889 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 50863.51 |
構造登録者 | |
主引用文献 | Melnick, M.,Mochalkin, I.,Lightle, S.,Narasimhan, L.,Mcdowell, L.,Sarver, R. Discovery and Initial Sar of Quinazoline Inhibitors of Glmu from Haemophilus Influenzae To be Published, |
実験手法 | X-RAY DIFFRACTION (1.99 Å) |
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