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2ILP

Clostridium botulinum Serotype A Light Chain inhibited by 4-chlorocinnamic hydroxamate

Summary for 2ILP
Entry DOI10.2210/pdb2ilp/pdb
DescriptorBotulinum neurotoxin A light-chain, ZINC ION, PHOSPHATE ION, ... (5 entities in total)
Functional Keywordsclostridium botulinum neurotoxin, type a, substrate specificity, substrate switching, protease inhibitors, hydrolase
Biological sourceClostridium botulinum
Total number of polymer chains2
Total formula weight102255.57
Authors
Silvaggi, N.R.,Allen, K.N. (deposition date: 2006-10-03, release date: 2007-06-05, Last modification date: 2024-02-21)
Primary citationSilvaggi, N.R.,Boldt, G.E.,Hixon, M.S.,Kennedy, J.P.,Tzipori, S.,Janda, K.D.,Allen, K.N.
Structures of Clostridium botulinum Neurotoxin Serotype A Light Chain Complexed with Small-Molecule Inhibitors Highlight Active-Site Flexibility.
Chem.Biol., 14:533-542, 2007
Cited by
PubMed: 17524984
DOI: 10.1016/j.chembiol.2007.03.014
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

217705

數據於2024-03-27公開中

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