2A0X
Structure of human purine nucleoside phosphorylase H257F mutant
Summary for 2A0X
Entry DOI | 10.2210/pdb2a0x/pdb |
Related | 1A0W 2A0Y |
Descriptor | Purine nucleoside phosphorylase, SULFATE ION, 7-[[(3R,4R)-3-(hydroxymethyl)-4-oxidanyl-pyrrolidin-1-ium-1-yl]methyl]-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one, ... (4 entities in total) |
Functional Keywords | purine nucleoside phosphorylase, transition state inhibitor, mutant, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 32651.32 |
Authors | Murkin, A.S.,Shi, W.,Schramm, V.L. (deposition date: 2005-06-17, release date: 2006-06-06, Last modification date: 2023-08-23) |
Primary citation | Murkin, A.S.,Birck, M.R.,Rinaldo-Matthis, A.,Shi, W.,Taylor, E.A.,Almo, S.C.,Schramm, V.L. Neighboring group participation in the transition state of human purine nucleoside phosphorylase. Biochemistry, 46:5038-5049, 2007 Cited by PubMed: 17407325DOI: 10.1021/bi700147b PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.28 Å) |
Structure validation
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