1QHI
HERPES SIMPLEX VIRUS TYPE-I THYMIDINE KINASE COMPLEXED WITH A NOVEL NON-SUBSTRATE INHIBITOR, 9-(4-HYDROXYBUTYL)-N2-PHENYLGUANINE
1QHI の概要
エントリーDOI | 10.2210/pdb1qhi/pdb |
分子名称 | PROTEIN (THYMIDINE KINASE), SULFATE ION, 9-(4-HYDROXYBUTYL)-N2-PHENYLGUANINE, ... (4 entities in total) |
機能のキーワード | transferase, transferase (phosphotransferase) thymidine, transferase (phosphotransferase) thymidine kinase; viridae; ds-dna enveloped viruses; herpesviridae; alphaherpesvirinae novel inhibitor |
由来する生物種 | Herpes simplex virus (type 1 / strain 17) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 80569.97 |
構造登録者 | Bennett, M.S.,Wien, F.,Champness, J.N.,Batuwangala, T.,Rutherford, T.,Summers, W.C.,Sun, H.,Wright, G.,Sanderson, M.R. (登録日: 1999-05-12, 公開日: 1999-07-09, 最終更新日: 2023-08-16) |
主引用文献 | Bennett, M.S.,Wien, F.,Champness, J.N.,Batuwangala, T.,Rutherford, T.,Summers, W.C.,Sun, H.,Wright, G.,Sanderson, M.R. Structure to 1.9 A resolution of a complex with herpes simplex virus type-1 thymidine kinase of a novel, non-substrate inhibitor: X-ray crystallographic comparison with binding of aciclovir. FEBS Lett., 443:121-125, 1999 Cited by PubMed: 9989588DOI: 10.1016/S0014-5793(98)01619-6 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.9 Å) |
構造検証レポート
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