1Q4L
GSK-3 Beta complexed with Inhibitor I-5
Summary for 1Q4L
Entry DOI | 10.2210/pdb1q4l/pdb |
Related | 1PYX 1Q3D 1Q3W 1Q41 |
Descriptor | GLYCOGEN SYNTHASE KINASE-3 BETA, 2-CHLORO-5-[4-(3-CHLORO-PHENYL)-2,5-DIOXO-2,5-DIHYDRO-1H-PYRROL-3-YLAMINO]-BENZOIC ACID (3 entities in total) |
Functional Keywords | kinase, insulin pathway, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: P49841 |
Total number of polymer chains | 2 |
Total formula weight | 94917.30 |
Authors | Bertrand, J.A.,Thieffine, S.,Vulpetti, A.,Cristiani, C.,Valsasina, B.,Knapp, S.,Kalisz, H.M.,Flocco, M. (deposition date: 2003-08-04, release date: 2003-10-14, Last modification date: 2023-08-16) |
Primary citation | Bertrand, J.A.,Thieffine, S.,Vulpetti, A.,Cristiani, C.,Valsasina, B.,Knapp, S.,Kalisz, H.M.,Flocco, M. Structural Characterization of the Gsk-3Beta Active Site Using Selective and Non-selective ATP-Mimetic Inhibitors J.Mol.Biol., 333:393-407, 2003 Cited by PubMed: 14529625DOI: 10.1016/j.jmb.2003.08.031 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.77 Å) |
Structure validation
Download full validation report