1CPU
SUBSITE MAPPING OF THE ACTIVE SITE OF HUMAN PANCREATIC ALPHA-AMYLASE USING SUBSTRATES, THE PHARMACOLOGICAL INHIBITOR ACARBOSE, AND AN ACTIVE SITE VARIANT
1CPU の概要
エントリーDOI | 10.2210/pdb1cpu/pdb |
関連するBIRD辞書のPRD_ID | PRD_900001 |
分子名称 | PROTEIN (ALPHA-AMYLASE), 4-amino-4,6-dideoxy-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... (8 entities in total) |
機能のキーワード | amylase, acarbose, glycosylation, mutagenesis, diabetes, catalysis, pancreatic, enzyme, human, hydrolase |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 57071.82 |
構造登録者 | Brayer, G.D.,Sidhu, G.,Maurus, R.,Rydberg, E.H.,Braun, C.,Wang, Y.,Nguyen, N.T.,Overall, C.M.,Withers, S.G. (登録日: 1999-06-07, 公開日: 1999-06-14, 最終更新日: 2023-12-27) |
主引用文献 | Brayer, G.D.,Sidhu, G.,Maurus, R.,Rydberg, E.H.,Braun, C.,Wang, Y.,Nguyen, N.T.,Overall, C.M.,Withers, S.G. Subsite mapping of the human pancreatic alpha-amylase active site through structural, kinetic, and mutagenesis techniques. Biochemistry, 39:4778-4791, 2000 Cited by PubMed: 10769135DOI: 10.1021/bi9921182 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2 Å) |
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