1BX6
CRYSTAL STRUCTURE OF THE POTENT NATURAL PRODUCT INHIBITOR BALANOL IN COMPLEX WITH THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE
1BX6 の概要
エントリーDOI | 10.2210/pdb1bx6/pdb |
分子名称 | CAMP-DEPENDENT PROTEIN KINASE, BALANOL (3 entities in total) |
機能のキーワード | serine/threonine-protein kinase, balanol, conformational changes, inhibition, protein kinase pka, serine-threonine-protein kinase complex |
由来する生物種 | Mus musculus (house mouse) |
細胞内の位置 | Cytoplasm (By similarity): P05132 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 41287.81 |
構造登録者 | Narayana, N.,Xuong, N.-H.,Ten Eyck, L.F.,Taylor, S.S. (登録日: 1998-10-13, 公開日: 1999-04-27, 最終更新日: 2023-08-09) |
主引用文献 | Narayana, N.,Diller, T.C.,Koide, K.,Bunnage, M.E.,Nicolaou, K.C.,Brunton, L.L.,Xuong, N.H.,Ten Eyck, L.F.,Taylor, S.S. Crystal structure of the potent natural product inhibitor balanol in complex with the catalytic subunit of cAMP-dependent protein kinase. Biochemistry, 38:2367-2376, 1999 Cited by PubMed: 10029530DOI: 10.1021/bi9820659 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.1 Å) |
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