6BKW
BTK complex with compound 12
エンティティ
Entity ID | 鎖名 | 説明 | 種類 | 鎖長 | 化学式量 | 分子数 | データベース名(アクセス番号) | 由来する生物種 | エンティティの一般名 |
1 | A | Tyrosine-protein kinase BTK | polymer | 287 | 33878.7 | 1 | UniProt (Q06187) Pfam (PF07714) In PDB | Homo sapiens (Human) | Agammaglobulinemia tyrosine kinase,ATK,B-cell progenitor kinase,BPK,Bruton tyrosine kinase |
2 | A | SULFATE ION | non-polymer | 96.1 | 3 | Chemie (SO4) | |||
3 | A | N-(3-{5-[(1,5-dimethyl-1H-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | non-polymer | 510.6 | 1 | Chemie (DXM) | |||
4 | A | triphenylphosphane | non-polymer | 262.3 | 1 | Chemie (FPZ) | |||
5 | A | GLYCEROL | non-polymer | 92.1 | 2 | Chemie (GOL) | |||
6 | water | water | 18.0 | 203 | Chemie (HOH) |
配列変更
A: 393 - 657 (UniProt: Q06187)
PDB | 外部データベース | 詳細 |
---|---|---|
Met 392 | - | initiating methionine |
Asn 658 | - | expression tag |
Leu 659 | - | expression tag |
Tyr 660 | - | expression tag |
Phe 661 | - | expression tag |
Gln 662 | - | expression tag |
Gly 663 | - | expression tag |
Glu 664 | - | expression tag |
Glu 665 | - | expression tag |
Tyr 666 | - | expression tag |
Met 667 | - | expression tag |
Pro 668 | - | expression tag |
Thr 669 | - | expression tag |
Glu 670 | - | expression tag |
His 671 | - | expression tag |
His 672 | - | expression tag |
His 673 | - | expression tag |
His 674 | - | expression tag |
His 675 | - | expression tag |
His 676 | - | expression tag |
His 677 | - | expression tag |
His 678 | - | expression tag |
配列ビューア
非対称単位の内容
タンパク質・ 核酸鎖 | 鎖の数 | 1 |
化学式量合計 | 33878.7 | |
タンパク質・ 核酸・ 糖鎖以外* | 分子数 | 7 |
化学式量合計 | 1245.2 | |
全て* | 化学式量合計 | 35123.9 |