4KHM
HCV NS5B GT1A with GSK5852
エンティティ
Entity ID | 鎖名 | 説明 | 種類 | 鎖長 | 化学式量 | 分子数 | データベース名(アクセス番号) | 由来する生物種 | エンティティの一般名 |
1 | A, B | HCV Polymerase | polymer | 579 | 64035.3 | 2 | UniProt (B1PPP0) Pfam (PF00998) In PDB | Hepatitis C virus subtype 1a (HCV) | RNA-directed RNA polymerase, NS5B, p68 |
2 | A, B | [4-({[5-cyclopropyl-2-(4-fluorophenyl)-3-(methylcarbamoyl)-1-benzofuran-6-yl](methylsulfonyl)amino}methyl)-2-fluorophenyl]boronic acid | non-polymer | 554.4 | 2 | Chemie (1PV) | |||
3 | A, B | SULFATE ION | non-polymer | 96.1 | 7 | Chemie (SO4) | |||
4 | water | water | 18.0 | 922 | Chemie (HOH) |
配列変更
A, B: 1 - 570 (UniProt: B1PPP0)
PDB | 外部データベース | 詳細 |
---|---|---|
Met 0 | - | expression tag |
Ser 5 | Thr 2425 | variant |
Val 11 | Ile 2431 | variant |
Tyr 101 | Phe 2521 | engineered mutation |
Ser 110 | Cys 2530 | engineered mutation |
Ser 113 | Arg 2533 | engineered mutation |
Arg 114 | Lys 2534 | engineered mutation |
Ala 546 | Asp 2966 | variant |
Leu 571 | - | expression tag |
Glu 572 | - | expression tag |
His 573 | - | expression tag |
His 574 | - | expression tag |
His 575 | - | expression tag |
His 576 | - | expression tag |
His 577 | - | expression tag |
His 578 | - | expression tag |
配列ビューア
非対称単位の内容
タンパク質・ 核酸鎖 | 鎖の数 | 2 |
化学式量合計 | 128070.7 | |
タンパク質・ 核酸・ 糖鎖以外* | 分子数 | 9 |
化学式量合計 | 1781.2 | |
全て* | 化学式量合計 | 129851.9 |