4BKZ
Crystal structure of unphosphorylated Maternal Embryonic Leucine zipper Kinase (MELK) in complex with a benzodipyrazole inhibitor
エンティティ
Entity ID | 鎖名 | 説明 | 種類 | 鎖長 | 化学式量 | 分子数 | データベース名(アクセス番号) | 由来する生物種 | エンティティの一般名 |
1 | A | MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE | polymer | 347 | 40220.5 | 1 | UniProt (Q14680) Pfam (PF00069) Pfam (PF21594) In PDB | HOMO SAPIENS (HUMAN) | HMELK, PROTEIN KINASE EG3, PEG3 KINASE, PROTEIN KINASE PK38, HPK38, TYROSINE-PROTEIN KINASE MELK |
2 | A | N-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | non-polymer | 369.4 | 1 | Chemie (1WS) | |||
3 | water | water | 18.0 | 80 | Chemie (HOH) |
配列変更
A: 2 - 340 (UniProt: Q14680)
PDB | 外部データベース | 詳細 |
---|---|---|
Gly 0 | - | expression tag |
Pro 1 | - | expression tag |
His 341 | - | expression tag |
His 342 | - | expression tag |
His 343 | - | expression tag |
His 344 | - | expression tag |
His 345 | - | expression tag |
His 346 | - | expression tag |
配列ビューア
非対称単位の内容
タンパク質・ 核酸鎖 | 鎖の数 | 1 |
化学式量合計 | 40220.5 | |
タンパク質・ 核酸・ 糖鎖以外* | 分子数 | 1 |
化学式量合計 | 369.4 | |
全て* | 化学式量合計 | 40589.9 |