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2OC0

Structure of NS3 complexed with a ketoamide inhibitor SCh491762

エンティティ
Entity ID鎖名説明種類鎖長化学式量分子数データベース名(アクセス番号)由来する生物種エンティティの一般名
1A, CHepatitis C Viruspolymer20021233.22UniProt (Q9ELS8)
Pfam (PF02907)
UniProt (by SIFTS) (P27958)
In PDB
Hepatitis C virus
2B, DHepatitis C viruspolymer232394.02UniProt (Q9QP06)
Pfam (PF01006)
UniProt (by SIFTS) (P27958)
In PDB
3A, CZINC IONnon-polymer65.42Chemie (ZN)
4ABETA-MERCAPTOETHANOLnon-polymer78.11Chemie (BME)
5ATERT-BUTYL {(1S)-2-[(1R,2S,5S)-2-({[(1S)-3-AMINO-1-(CYCLOBUTYLMETHYL)-2,3-DIOXOPROPYL]AMINO}CARBONYL)-6,6-DIMETHYL-3-AZABICYCLO[3.1.0]HEX-3-YL]-1-CYCLOHEXYL-2-OXOETHYL}CARBAMATEnon-polymer546.71Chemie (HU1)
6waterwater18.0210Chemie (HOH)
配列変更
A, C: 1 - 181 (UniProt: Q9ELS8)
PDB外部データベース詳細
Met -10-cloning artifact
Ala -9-cloning artifact
Ser -8-cloning artifact
Met -7-cloning artifact
Thr -6-cloning artifact
Gly -5-cloning artifact
Gly -4-cloning artifact
Gln -3-cloning artifact
Gln -2-cloning artifact
Met -1-cloning artifact
Gly 0-cloning artifact
Arg 119Gln 1145conflict
Gly 182-cloning artifact
Ser 183-cloning artifact
His 184-expression tag
His 185-expression tag
His 186-expression tag
His 187-expression tag
His 188-expression tag
His 189-expression tag
B, D: 21 - 39 (UniProt: Q9QP06)
PDB外部データベース詳細
Lys 19-cloning artifact
Lys 20-cloning artifact
Lys 40-cloning artifact
Lys 41-cloning artifact
配列ビューア
非対称単位の内容
タンパク質・
核酸鎖
鎖の数4
化学式量合計47254.5
タンパク質・
核酸・
糖鎖以外*
分子数4
化学式量合計755.6
全て*化学式量合計48010.2
*水分子は含んでいません

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件を2024-09-18に公開中

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